VASG Alfaxalone | 動物用藥查詢網
![VASG Alfaxalone](https://i.imgur.com/TbfVXFL.jpg)
I.M.sedation.alfaxalone.midazolam;Dog/cat.2–4mg/kg(1–2mg/lb).0.3mg/kg(0.15mg/lb) ...
![VASG Alfaxalone](https://i.imgur.com/TbfVXFL.jpg)
Alfaxalone is not a new drug. It was originally introduced in the 1970s as a mixture with alfadolone. The brand names were Althesin® for the human product and Saffan® for the veterinary market. Both products were withdrawn from the market because of severe adverse effects. These adverse effects (histamine release and anaphylactic reactions) were very probably caused by the solubilising agent Cremophor EL®, a derivate of castor oil.
Alfaxalone is remarketed as a water-soluble neuroanaesthetic. Water solubility was achieved by binding the alfaxalone-molecule to a cyclodextrine molecule. It is rapidly metabolized by the liver and does not cause histamine release like the former formulation. Alfaxalone’s anaesthetic action is due to its binding to GABA-receptors.
With the introduction of Alfaxan® veterinarians have access to another anesthetic with a ...
Alfaxalone for Anesthesia in Dogs and Cats | 動物用藥查詢網
Alfaxalone | 動物用藥查詢網
Alfaxan | 動物用藥查詢網
Comparison of the sedative effects of alfaxalone and ... | 動物用藥查詢網
Intramuscular use of alfaxalone in dogs | 動物用藥查詢網
The anesthetic effects of intramuscular alfaxalone in dogs ... | 動物用藥查詢網
VASG Alfaxalone | 動物用藥查詢網
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