DORIBAX® (doripenem) powder | 動物用藥查詢網
![DORIBAX® (doripenem) powder](https://i.imgur.com/TbfVXFL.jpg)
2018年4月21日—Dosageandadministration;>50,Nodosageadjustmentnecessary;≥30to≤50,250mg*administeredintravenously(over1hour)every8hours.
![DORIBAX® (doripenem) powder](https://i.imgur.com/TbfVXFL.jpg)
Doripenem is a carbapenem with in vitro antibacterial activity against aerobic and anaerobic Gram-positive and Gram-negative bacteria.
Mechanism of Action Doripenem is an antibacterial drug. Microbiology Doripenem belongs to the carbapenem class of antimicrobials. Doripenem exerts its bactericidal activity by inhibiting bacterial cell wall biosynthesis. Doripenem inactivates multiple essential penicillin-binding proteins (PBPs) resulting in inhibition of cell wall synthesis with subsequent cell death. In E. coli and P. aeruginosa, doripenem binds to PBP 2, which is involved in the maintenance of cell shape, as well as to PBPs 3 and 4.
Mechanism(s) of Resistance Bacterial resistance mechanisms that affect doripenem include drug inactivation by carbapenem-hydrolyzing enzymes, mutant or acquired PBPs, decreased outer membrane permeability and active efflux. ...
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